氯化钾的应用?
250ml盐水中加了7.5ml氯化钾,还能再加门冬氨酸钾镁针吗?
推荐回答(2个)
别名:氯化钾
药理作用: 正常人体内总钾量平均为120g,其中仅约2%存在于细胞外液,其余几乎集中在细胞内。钾为细胞内主要阳离子,是维持细胞内渗透压的重要成分。钾通过与细胞外的氢离子交换参与酸硷平衡的调节,当体内缺钾时,细胞内钾离子外移而细胞外氢、钠离子内移,其结果为细胞内酸中毒,血钾过高时则相反。钾参与糖、蛋白质的合成及二磷酸腺苷转化为三磷酸腺苷的能量代谢。钾也参与神经冲动传导和神经末梢递质乙酰胆碱的合成。缺钾对心肌兴奋性增高,钾过多时则抑制心肌的自律性、传导性和兴奋性。因而钾浓度变化影响洋地黄对心脏的作用。当钾摄入量不足,排出量增多或在体内分布异常可引起低钾血症。服药后1小时,病人血清钾显著升高,第2小时血钾继续上升至接近血钾最高限。第1小时溶出度为12.5%,第2小时为23.5%,服本药2g后1小时,消化道中有钾,3.325mEq,第2小时内共有6.25mEq钾可被吸收。若以病人体重为50kg计算,第1小时可提高血钾浓度1.6mmol/L,第2小时可提高3.1mmol/L。肾功能正常而又有正常尿量的人,口服常量钾盐不可能导致高血钾症。血钾浓度持续保持在较高水平至12小时后才下降。他药后6-8小时,尿排钾量逐渐增加。控释片的药物浓度达峰时间较氯化钾溶液迟,药时曲线下面积较大,相对生物利用度为溶液组的111.3%。控释片在消化道中缓慢溶出氯化钾,被吸收后保持较稳定的血钾浓度,因而提高了生物利用度。每日2次给药可有较防止长期利尿所致的低血钾,特别适合重症或需长期服药的患者。
适应症: 用于低钾血症(多由严重吐泻不能进食、长期应用排钾利尿剂或肾上腺皮质激素所引起)的防治,亦可用于强心甙中毒引起的阵发性心动过速或频发室性期外收缩。本药为电解质补充剂,以及洋地黄中毒引起的心律失常。亦可做为利尿的辅助剂。
用法用量: 补充钾盐大多采用口服,1次1g,1日3次。血钾过低,病情危急或吐泻严重口服不易吸收时,可用静滴,每次用10%~15%液10ml,用5%~10%葡萄糖液500ml稀释或根据病情酌定用量。应在心电图密切监视下进行,如出现高钾血症,则立即停用。口服:氯化钾1~2g,3~4次/d。成人每日早晚各服2片。
不良反应: 口服对胃肠道有刺激性,可出现恶心、呕吐、腹泻。故宜用缓释片或配成10%呤液于饭后服用以减少刺激性。氯化钾不可肌注或静注给予。静滴时必须先用5%葡萄糖注射液稀释至0.2%~0.4%,滴注速度应缓慢,一般每小时不超过氯化钾1g,否则可抑制心脏功能。如出现心脏毒性可缓缓静注10%葡萄糖酸钙10~20m1,并静滴含胰岛素的5%葡萄糖注射液(2g葡萄糖需:单位胰岛素)解救。肾功能不全、肾上腺皮质功能不全、急性脱水等患者慎用,无尿时禁用,以免引起高钾其症。
注意事项: (1)静滴过量时可出现疲乏,肌张力减低、反射消失、周围循环衰竭、心率减慢甚至心脏停搏。(2)肾功能严重减退者尿少时慎用,无尿或血钾过高时忌用。(3)脱水病例一般先给不含钾的液体(也可给复方氯化钾液,因其含钾浓度低,不致引起高钾血症),等排尿后再补钾。(4)静滴时,速度宜慢,溶液不可太浓(一般不超过0.2%~0.4%,治疗心律失常时可加至0.6%~(0.7%),否则不仅引起局部剧痛,且可导致心脏停搏。 (5)口服本品溶液或无糖衣片,对胃肠道有较强的刺激性,部分病人难以耐受。当病人服后出现腹部不适、疼痛等症状时,应加警惕,因服用氯化钾片等制剂时,有造成胃肠溃疡、坏死或狭窄等并发症的可能,宜采用本品的10%水溶液稀释于饮料中在餐后服用,以减少刺激性。如有氯化钾控释片供用则更好。肾功能不全者慎用。 [禁忌]少尿和尿闭者
规格:片剂:每片0.25g;0.5g。控释片(SLOwK):每片0.6g。微囊片(PEL一K):每片0.75g。注射液:每支1g(10ml)。复方氯化钾注射液:内含氯化钾0.28%、氯化钠 0.42%及乳酸钠0.63%,可用于代谢性酸血症及低血钾。用量视病情而定,一般每日量500~1000ml,静滴。
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